產品描述: IDO-IN-7 (NLG-919 analogue) is a a potent IDO1 inhibitor with an IC50 of 38 nM. |
靶點:
IDO1:38 nM (IC50);Indoleamine2,3-Dioxygenase(IDO) |
參考文獻:
1. Coletti A, et al. Fragment-based approach to identify IDO1 inhibitor building blocks. Eur J Med Chem. 2017 Dec 1;141:169-177. |
溶解性:
DMSO : 50 mg/mL (177.07 mM; Need ultrasonic) Ethanol : 25 mg/mL (88.53 mM; Need ultrasonic) |
保存條件:
-20℃ |
配置溶液濃度參考:
|
1mg |
5mg |
10mg |
1 mM |
3.541 ml |
17.707 ml |
35.413 ml |
5 mM |
0.708 ml |
3.541 ml |
7.083 ml |
10 mM |
0.354 ml |
1.771 ml |
3.541 ml |
50 mM |
0.071 ml |
0.354 ml |
0.708 ml |
|
注意: |
部分產品我司僅能提供部分信息,我司不保證所提供信息的權威性,僅供客戶參考交流研究之用。 |